Cas No. |
Product name |
1370261-97-4 |
PRT062607 (P505-15 HCL) |
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PRT062607 (P505-15) HCl is a novel, highly selective Syk inhibitor with IC50 of 1 nM, >80-fold selective for Syk than Fgr, Lyn, FAK, Pyk2 and Zap70 |
860352-01-8 |
AZD7762 |
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AZD7762 is a potent and selective inhibitor of Chk1 with IC50 of 5 nM. It is equally potent against Chk2 and less potent against CAM, Yes, Fyn, Lyn, Hck and Lck. Phase 1 |
658084-64-1 |
FK866 |
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APO866 effectively inhibits nicotinamide phosphoribosyltransferase (NMPRTase) with IC50 of 0.09 nM. Phase 1/2 |
841205-47-8 |
MK-2866 (GTx-024) |
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MK-2866 (GTx-024) is a selective androgen receptor modulator (SARM) with Ki of 3.8 nM, and is tissue-selective for anabolic organs. Phase 3 |
401900-40-1 |
Andarine |
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Andarine is a selective non-steroidal androgen receptor (AR) agonist with Ki of 4 nM, tissue-selective for anabolic organs |
162831-31-4 |
IEM1754 |
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IEM 1754 dihydrobroMide is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM |
1240299-33-5 |
AZD3514 |
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AZD3514 is a potent and oral androgen receptor downregulator with Ki of 2.2 μM and has ability of reducing AR protein expression |
856925-71-8 |
(-)-Blebbistatin |
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(-)-Blebbistatin is a cell-permeable inhibitor for non muscle myosin II ATPase with IC50 of ~2 μM, does not inhibit myosin light chain kinase, inhibits contraction of the cle... |
1009119-64-5 |
Daclatasvir (BMS790052) |
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BMS-790052 is a highly selective inhibitor of HCV NS5A with EC50 of 9-50 pM, for a broad range of HCV replicon genotypes and the JFH-1 genotype 2a infectious virus in cell cu... |
1338466-77-5 |
EPZ004777 |
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EPZ004777 is a potent, selective DOT1L inhibitor with IC50 of 0.4 nM |